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  4. Derivatives of (2R,3R,4S)-2-Aminomethylpyrrolidine-3,4-diol are Selective alpha-Mannosidase Inhibitors
 
research article

Derivatives of (2R,3R,4S)-2-Aminomethylpyrrolidine-3,4-diol are Selective alpha-Mannosidase Inhibitors

Popowycz, Florence  
•
Gerber-Lemaire, Sandrine  
•
Demange, Raynald  
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2001
Bioorganic and Medicinal Chemistry Letters

A collection of (2R,3R,4S)-3,4-dihydroxypyrrolidin-2-yl derivatives have been tested for their inhibitory activities toward 25 glycosidases. Competitive (K-i=7.4 VM) and selective inhibition of alpha -mannosidase from jack bean has been found for (2R,3R,4S)-2-[(benzylamino)methyl]pyrrolidine-3,4-diol and other derivatives.

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Type
research article
DOI
10.1016/S0960-894X(01)00477-2
Author(s)
Popowycz, Florence  
•
Gerber-Lemaire, Sandrine  
•
Demange, Raynald  
•
Rodriguez-Garcia, Eliaizar  
•
Carmona Asenjo, Ana Teresa  
•
Robina, Inmaculada
•
Vogel, Pierre  
Date Issued

2001

Published in
Bioorganic and Medicinal Chemistry Letters
Volume

11

Issue

18

Start page

2489

End page

2493

Subjects

3 deoxy derivatives

•

mannostatin-a

•

glycosidase inhibitors

•

biological-activities

•

advanced malignancies

•

processing inhibitor

•

class-i

•

swainsonine

•

thioglycoside

•

disaccharides

Editorial or Peer reviewed

REVIEWED

Written at

EPFL

EPFL units
LGSA  
Available on Infoscience
June 8, 2006
Use this identifier to reference this record
https://infoscience.epfl.ch/handle/20.500.14299/230378
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