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research article
Synthesis of polycyclic aminal heterocycles via decarboxylative cyclisation of dipeptide derivatives
February 15, 2022
An oxidative-decarboxylative intramolecular cyclisation of dipeptide derivatives is reported. This transformation is promoted by phenyl iodine(iii) diacetate (PIDA) in combination with BF3 center dot OEt2. The reaction gives access to a variety of valuable polycyclic N-heterocyclic scaffolds containing 5-, 6-, or 7-membered rings.
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Name
CC2022-3473-GreenAccess1.pdf
Type
Preprint
Access type
openaccess
License Condition
CC BY
Size
10.51 MB
Format
Adobe PDF
Checksum (MD5)
7e24350f3ab7e3bddf3c5bebc0bf13ae
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Name
CC2022-3473-GreenAccess.pdf
Type
Postprint
Access type
embargo
Embargo End Date
2023-02-15
License Condition
CC BY
Size
10.52 MB
Format
Adobe PDF
Checksum (MD5)
49b57bfd01a583b3e167d9cb061f15ab