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research article
Enantioselective palladium(0)-catalyzed intramolecular cyclopropane functionalization: access to dihydroquinolones, dihydroisoquinolones and the BMS-791325 ring system
2015
Taddol-based phosphoramidite ligands enable enantioselective palladium(0)-catalyzed C-H arylation of cyclopropanes. The cyclized products are obtained in high yields and enantioselectivities. The reported method provides efficient access to a broad range of synthetically attractive cyclopropyl containing dihydroquinolones and dihydroisoquinolones as well as allows for an efficient enantioselective construction of the 7-membered ring of the cyclopropyl indolobenzazepine core of BMS-791325.
Type
research article
Web of Science ID
WOS:000359214100009
Authors
Publication date
2015
Publisher
Published in
Volume
6
Issue
9
Start page
5164
End page
5171
Peer reviewed
REVIEWED
EPFL units
Available on Infoscience
September 28, 2015
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