A reaction of 2-acyl substituted tetrahydroquinolines, prepared by Lewis acid-catalyzed three-component reaction of α-oxo aldehydes, anilines, and dienophiles, with in situ generated arynes afforded 5,6-dihydroindolo[1,2-a]- quinolines in good to excellent yields.
Titre
Three-Component Povarov Reaction–Heteroannulation with Arynes: Synthesis of 5,6-Dihydroindolo[1,2‑a]quinolines
Publié dans
Organic Letters
Pagination
4
Volume
16
Numéro
6
Pages
1756-1759
Date
2014
Editeur
Washington, Amer Chemical Soc
ISSN
1523-7052
Date de création de la notice
2014-03-22
