Synthesis of Indoles by Copper-Catalyzed Heteroannulation of o-Aminophenylboronic Acid Pinacol Esters with β-Keto Esters

Copper-catalyzed coupling of ortho-aminophenylboronic acid pinacol esters with β-ketoesters afforded, under mild base-free oxidative conditions, 2,3-disubstituted indoles featuring a key Chan-Lam type carbon-carbon bond forming reaction.


Published in:
Synthesis, 44, 24, 3811-3814
Year:
2012
Publisher:
Stuttgart, Georg Thieme Verlag Kg
ISSN:
1437-210X
Keywords:
Laboratories:




 Record created 2012-12-09, last modified 2018-12-03


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