2-homopiperazine-1-yl-4h-1,3-benzothiazine-4-one derivatives and process for the preparation of 2- (homo)piperazine 1,3-benzothiazine-4-one hydrochlorides
2-homopiperazine-1-yl-4H-l, 3 -bensothiazine-4-one derivatives of formula (I) are provided. They are useful in the treatment of bacterial infections, in particular tuberculosis, buruli ulcer and leprosy. A process for the preparation of 2- (homo)piperazine 1, 3-benzothiazine-4-one hydrochlorides is also provided.
52780412
Alternative title(s) : (de) 2-homopiperazin-1-yl-4h-1,3-benzothiazin-4-on-derivate und verfahren zur herstellung von 2-(homo)piperazin 1,3-benzothiazin-4-on-hydrochloriden (fr) Dà rivés de 2-homopipérazine-1-yl-4h-1,3-benzothiazine-4-one et procédé pour la préparation d'hydrochlorures de 2- (homo) pipérazine 1,3-benzothiazine-4-one (en) 2-homopiperazine-1-yl-4h-1,3-benzothiazine-4-one derivatives and process for the preparation of 2-(homo)piperazine 1,3-benzothiazine-4-one hydrochlorides
TTO:6.1036
| DOI | Country code | Kind code | Date issued |
ES2905453 | ES | T3 | 2022-04-08 |
PL3274339 | PL | T3 | 2022-03-07 |
EP3919480 | EP | A1 | 2021-12-08 |
EP3274339 | EP | B1 | 2021-10-13 |
UA123724 | UA | C2 | 2021-05-26 |
GEP20217258 | GE | B | 2021-05-25 |
CN107567439 | CN | B | 2021-04-16 |
EA035946 | EA | B1 | 2020-09-04 |
EA202091353 | EA | A1 | 2020-08-19 |
GEP20207127 | GE | B | 2020-06-25 |
US10358442 | US | B2 | 2019-07-23 |
US2019077798 | US | A1 | 2019-03-14 |
US10160754 | US | B2 | 2018-12-25 |
EA201792095 | EA | A1 | 2018-03-30 |
US2018051016 | US | A1 | 2018-02-22 |
EP3274339 | EP | A1 | 2018-01-31 |
CN107567439 | CN | A | 2018-01-09 |
CA2980653 | CA | A1 | 2016-09-29 |
WO2016151011 | WO | A1 | 2016-09-29 |
EP3072889 | EP | A1 | 2016-09-28 |